-2012-

Synthesis of two neurokinin NK1 receptor receptor antagonists : (+)-L-733,060 and (-)-L-733,061. A. Cochi, D. Gomez Pardo, J. Cossy Heterocycles 2012, 86, 89-116.

Efficient synthesis of substituted 3-azabicyclo[3.1.0]hexan-2-ones from 2-iodocyclopropanecarboxamides using a copper-free sonogashira coupling. B. de Carne-Carnavalet, A. Archambeau, C. Meyer, J. Cossy, B. Folleas, J.-L. Brayer, J.-P. Demoute Chemistry - A Eur. J. 2012, 18, 16716-16727.

Stereoselective synthesis of conjugated trienols from allylic alcohols and 1-iodo-1,3-dienes. D. Brandt, V. Bellosta, J. Cossy Org. Lett. 2012, 14, 5594-5597.

Fluorine as a regiocontrol element in the ring opening of bicyclic aziridiniums. Y. H. Lam, K. N. Houk, J. Cossy, D. Gomez Pardo, A. Cochi Helv. Chim. Acta 2012, 95, 2265-2277.

Two-step one-pot synthesis of benzoannulated spiroacetals by Suzuki-Miyaura coupling/acid-catalyzed spiroacetalization. A. N. Butkevich, A. Corbu, L. Meerpoel, I. Stansfield, P. Angibaud, P. Bonnet, J. Cossy, Janine Org. Lett. 2012, 14, 4998-5001.

[388] DNA as a tool for molecular discovery. M. Smietana, J.-J. Vasseur, J. Cossy, S. Arseniyadis in Modern Tools for the Synthesis of Complex Bioactive Molecules John Wiley & Sons, Inc., Hoboken, N. J. Edited by J. Cossy, S. Arseniyadis 2012, 539-555.

Formal synthesis of dictyostatin and synthesis of two dictyostatin analogues. J. Gallon, J. Esteban, S. Bouzbouz, M. Campbell, S. Reymond, J. Cossy Chemistry - A Eur. J. 2012, 18, 11788-11797.

First intramolecular alkylation of nitriles with primary and secondary alcohols catalyzed by iridium complexes. B. Anxionnat, D. Gomez Pardo, G. Ricci, J. Cossy Eur. J. Org. Chem. 2012, 4453-4456.

Ring expansion of cyclic beta-amino alcohols induced by diethylaminosulfur trifluoride : Synthesis of cyclic amines with a tertiary fluorine at C3. B. Anxionnat, B. Robert, P. George, G. Ricci, M.-A. Perrin, D. Gomez Pardo, J. Cossy J. Org. Chem. 2012, 77, 6087-6099.

Gold(I)-catalysed cycloisomerisation of 1,6-cyclopropene-enes. F. Miege, C. Meyer, J. Cossy Chemistry - A Eur. J. 2012, 18, 7810-7822.

Synthesis of amines from alcohols in a nonepimerizing one-pot sequence - Synthesis of bioactive compounds : cinacalcet and dexoxadrol. C. Guerin, V. Bellosta, G. Guillamot, J. Cossy Eur. J. Org. Chem. 2012, 2990-3000.

Access to optically active 3-aminopiperidines by ring expansion of prolinols : Thermodynamic versus kinetic control. A. Cochi, D. Gomez Pardo, J. Cossy Eur. J. Org. Chem. 2012, 2023-2040.

(E)-Dimethyl 2-oxopent-3-enylphosphonate : An excellent substrate for cross-metathesis - easy access to functionalized heterocycles. T. Cochet, D. Roche, V. Bellosta, J. Cossy Eur. J. Org. Chem. 2012, 801-809.

Catalytic diastereoselective reduction of alpha,beta-epoxy and alpha,beta-aziridinyl ynones. V. Druais, C. Meyer, J. Cossy Org. Lett. 2012 14, 516-519.

Total synthesis of nominal lyngbouilloside aglycon. A. ElMarrouni, R. Lebeuf, J. Gebauer, M. Heras, S. Arseniyadis, J. Cossy Org. Lett. 2012 14, 314-317.

Highly Efficient Stereoselective Catalytic C(sp3)-H Insertions with Donor Rhodium Carbenoids Generated from Cyclopropenes. A. Archambeau, F. Miege, C. Meyer, J. Cossy Angew. Chem., Int. Ed. 2012 51, 11540-11544.

Diastereoselective synthesis of the C17-C30 fragment of amphidinol 3. N. Rival, D. Hazelard, G. Hanquet, T. Kreuzer, C. Bensoussan, S. Reymond, J. Cossy, F. Colobert Org. Biomol. Chem. 2012 10, 9418-9428.

Diastereoselective metal-catalyzed synthesis of C-aryl and C-vinyl glycosides. L. Nicolas, P. Angibaud, I. Stansfield, P. Bonnet, L. Meerpoel, S. Reymond, J. Cossy Angew. Chem., Int. Ed. 2012, 51, 11101-11104.

Rhodium(III)-catalyzed allylic C-H bond amination. Synthesis of cyclic amines from omega-unsaturated N-sulfonylamines. T. Cochet, V. Bellosta, D. Roche, J.-Y. Ortholand, A. Greiner, J. Cossy Chem. Commun. 2012, 48, 10745-10747.

Catalysis-based enantioselective total synthesis of myxothiazole Z, (14S)-melithiazole G and (14S)-cystothiazole F. A. Colon, T. J. Hoffman, J. Gebauer, J. Dash, J. H. Rigby, S. Arseniyadis, J. Cossy Chem. Commun. 2012, 48, 10508-10510.

Kinetic resolution of propargylamines via a highly enantioselective non-enzymatic N-acylation process. A. Kolleth, S. Christoph, S. Arseniyadis, J. Cossy Chem. Commun. 2012, 48, 10511-10513.

A modular and scalable one-pot synthesis of polysubstituted furans. J. Fournier, S. Arseniyadis, J. Cossy Angew. Chem., Int. Ed. 2012, 51, 7562-7566.

Synthesis and evaluation of new polyenic compounds as potential PPARs modulators. D. Amans, V. Bellosta, C. Dacquet, A. Ktorza, N. Hennuyer, B. Staels, D.-H. Caignard, J. Cossy Org. Biomol. Chem. 2012, 10, 6169-6185.

Spiroketals : Toward the synthesis of 39-oxobistramide K. M. Commandeur, C. Commandeur, J. Cossy Pure and Applied Chemistry 2012, 84, 1567-1574.

Ritter reaction : Recent catalytic developments. A. Guérinot, S. Reymond, J. Cossy Eur. J. Org. Chem. 2012, 19-28.